Tandem hydroformylation/Fischer indole synthesis: a novel and convenient approach to indoles from olefins.
نویسندگان
چکیده
[reaction: see text] A novel one-pot synthesis of indole systems via tandem hydroformylation/Fischer indole synthesis starting from olefins and arylhydrazines is described. This tandem procedure leads directly to 3-substituted indoles if unsubstituted phenylhydrazine is used and to 3,5- respectively 3,7-disubstituted indoles if para- or ortho-substituted arylhydrazines are used.
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ورودعنوان ژورنال:
- Organic letters
دوره 5 18 شماره
صفحات -
تاریخ انتشار 2003